TG 4-155
| Overview | |
| Catalog # | bs-82326c-5-mg |
| Product Name | TG 4-155 |
| Specifications | |
| Storage Buffer | Off-white solid |
| Storage Condition | -20°C |
| Target | |
| Product Information | Potent and selective prostaglandin EP2 receptor antagonist, KB = 2.4 and 34.5 nM for EP2 and DP1 receptors respectively. Displays >500-fold selectivity for EP2 over other prostanoid receptors.1 Inhibits butaprost-induced proinflammatory cytokine production, cell proliferation and invasion of PC-3 cells in vitro.2 Inhibits PGE2-induced inflammatory response and may represent a novel pharmacologic intervention for tumorigenesis resulting from inflammation.1 |
| Description | CAS Number: 1164462-05-8 Chemical Name: (2E)-N-[2-(2-Methyl-1H-indol-1-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)-2-propenamide Molecular weight: 394.47 Formula: C23H26N2O4 Solubility: DMSO (35 mg/ml) Ethanol (10 mg/ml) Physical Properties: Off-white solid Purity: 98% by TLC, NMR (Conforms) |
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