GSK6853

Overview
Catalog #	bs-82758c-5-mg
Product Name	GSK6853
Specifications
Storage Buffer	Off-white solid
Storage Condition	-20°C
Target
Product Information	Very potent (pIC50 = 8.6 vs full length protein, 7.7 in cellular assays) inhibitor of Bromodomain and PHD Finger-containing 1 (BRPF1). It displayed >1600-fold selectivity over other bromodomains.
Description	CAS Number: 1910124-24-1 Chemical Name: N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide Molecular weight: 409.49 Formula: C22H27N5O3 Solubility: DMSO (25 mg/ml); ethanol (25 mg/ml) Physical Properties: White solid Purity: 98% by HPLC NMR (Conforms)