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TGN-020

Overview
Catalog # bs-80331C
Product Name TGN-020
Specifications
Storage Buffer powder
Storage Condition RT
Target
Product Information Molecular Weight:206.22

Formula:C8H6N4OS

Purity:>98%

Solubility:Soluble in DMSO (up to 10 mg/ml with warming)

Chemical Name:N-1,3,4-thiadiazol-2-yl-3-pyridinecarboxamide

Description Aquaporin 4 channel blocker, IC50 = 3.1 μM.1 Reduces ischemic cerebral edema in a mouse model of focal cerebral ischemia using MRI.2 Increases regional cerebral blood flow as determined in wild-type and AQP-4 knockout mice.3 Reduces brain edema when administered after onset of ischemia in rat models.4