Ki-16425
Overview | |
Catalog # | bs-1050c-2mg-solid |
Product Name | Ki-16425 |
Specifications | |
Storage Buffer | Powder |
Storage Condition | Store in dry, dark place at -20C for 1 year. |
Target | |
Product Information | Molecular Weight: 474.96 Formula: C23 H23 Cl N2 O5 S CAS Number: 355025-24-0 InChi Key: LLIFMNUXGDHTRO-UHFFFAOYSA-N InChi: InChI=1S/C23H23ClN2O5S/c1-14-21(25-23(29)30-15(2)18-5-3-4-6-19(18)24)22(31-26-14)17-9-7-16(8-10-17)13-32-12-11-20(27)28/h3-10,15H,11-13H2,1-2H3,(H,25,29)(H,27,28) Smiles: CC1=NOC(=C1NC(=O)OC(C)C1C=CC=CC=1Cl)C1C=CC(CSCCC(O)=O)=CC=1 Purity: 98.0 Solubility: 10 mM in DMSO Appearance: Solid Power. Shelf Life: 1.0 years |
Description | Ki16425 is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively, shows no activity at LPA4, LPA5, LPA6. IC50 value: 0.3/6.5/0.93 uM(Ki, LPA1/2/3) Target: LPA1/2/3 |