DJ-V 159
Overview | |
Catalog # | bs-82694c-5-mg |
Product Name | DJ-V 159 |
Specifications | |
Storage Buffer | White solid |
Storage Condition | RT |
Target | |
Product Information | GPRC6A is the receptor for osteocalcin as well as structurally unrelated ligands including L-amino acids, cations and anabolic steroids.1 GPRC6A is a potential therapeutic target for treating type 2 diabetes.2 DJ-V 159 is an agonist at GPRC6A which activates ERK and upregulates cAMP levels in HEK-193 cells expressing GPRC6A It stimulates insulin secretion in mouse -cells and lowers blood glucose in mouse models.3 |
Description | CAS Number: 2253744-53-3 Chemical Name: N1,N3-Bis(4-cyano-3-(trifluoromethyl)phenyl)isophthalamide Molecular weight: 502.37 Formula: C24H12F6N4O2 Solubility: DMSO (60 mg/ml) Physical Properties: Off-white solid Purity: 98% by TLC NMR (Conforms) |