RVX-208
Overview | |
Catalog # | bs-82278c-5-mg |
Product Name | RVX-208 |
Specifications | |
Storage Buffer | Light brown solid |
Storage Condition | -20°C |
Target | |
Product Information | RVX-208 is a potent BET bromodomain antagonist with IC50 of 0.510 μM for BD2, with approximately 170-fold selectivity over BD11,2. Increases apolipoprotein A-1 and HDL cholesterol in vitro and in vivo3. Reduces atherosclerosis4. |
Description | CAS Number: 1044870-39-4 Chemical Name: 2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-4(3H)-quinzolinone Molecular weight: 370.41 Formula: C20H22N2O5 Solubility: DMSO (75 mg/ml) Ethanol (4 mg/ml) Physical Properties: White solid Purity: 98% by TLC, NMR (Conforms) |