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Efaroxan HCl

Overview
Catalog # bs-82189c-50-mg
Product Name Efaroxan HCl
Specifications
Storage Buffer Pale yellow solid. (MP = 170-174°C)
Storage Condition -20°C
Target
Product Information Selective α2-adrenergic receptor antagonist1 (selectivity ratio of α2/α1 = 724)4 and imidazoline receptor antagonist2. Induces release of insulin in the rat insulinoma cell line RIN-5AH by interaction with ATP-sensitive potassium channels independently from imidazoline I1 or I2 receptors.3 Increases resting plasma insulin levels and markedly potentiates the rise in insulin levels produced by adrenaline in the rat.4
Description CAS Number: 89197-00-2

Chemical Name: 2-Ethyl-2-(imidazolin-2-yl)-2,3-dihydrobenzofuran, hydrochloride

Molecular weight: 252.74

Formula: C13H16N2O HCl

Solubility: Water (25 mg/ml)

Physical Properties: White solid

Purity: 98% by TLC, NMR (Conforms)