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BCTC

Overview
Catalog # bs-82058c-10-mg
Product Name BCTC
Specifications
Storage Buffer Off-white solid
Storage Condition RT
Target
Product Information Vanilloid receptor I (TRPV1) antagonist, IC50 = 35 nM for capsaicin-induced and 6 nM for acid-induced TRPV1 activation. Displays analgesic activity in rat models of neuropathic pain. Orally active and cell permeable.
Description CAS Number: 393514-24-4

Chemical Name: 4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide

Molecular weight: 372.9

Formula: C20H25ClN4O

Solubility: DMSO (25 mg/ml) Ethanol (15 mg/ml)

Physical Properties: Off-white solid

Purity: 98% by TLC [ 2% CH3OH in CH2Cl2; Rf = 0.25] NMR Conforms