DMU-2105
Overview | |
Catalog # | bs-7005c-10mg-solid |
Product Name | DMU-2105 |
Specifications | |
Storage Buffer | Powder |
Storage Condition | Store in dry, dark place at -20C for 1 year. |
Target | |
Product Information | Molecular Weight: 259.3 Formula: C18 H13 N O CAS Number: 1031063-36-1 InChi Key: VWBDGXJRQZDLRV-CSKARUKUSA-N InChi: InChI=1S/C18H13NO/c20-18(17-6-3-11-19-13-17)10-8-14-7-9-15-4-1-2-5-16(15)12-14/h1-13H/b10-8+ Smiles: O=C(C=CC1=CC2=CC=CC=C2C=C1)C1C=NC=CC=1 Purity: 98.0 Solubility: Soluble in DMSO Appearance: Solid Power Shelf Life: 1.0 years |
Description | DMU-2105 is a potent and selective CYP1B1 inhibitor with IC50s of 10 nM and 742 nM for CYP1B1 and CYP1A1, respectively. DMU-2105 showed a very high level of selectivity towards CYP1B1 with respect to the IC50 values obtained with CYP1A1, CYP1A2, CYP3A4, CYP2D6, CYP2C9 and CYP2C19 Sacchrosomes™. |