AM251

Overview
Catalog #	bs-80370C
Product Name	AM251
Specifications
Storage Buffer	powder
Storage Condition	-20°C
Target
Product Information	Molecular Weight:555.24 Formula:C22H21Cl2IN4O Purity:>98% Solubility:Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 13 mg/ml) Chemical Name:N-(Piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide
Description	A potent cannabinoid CB1 receptor antagonist with selectivity over CB2 receptors (306-fold).1-3 Displays anorectic effects and antidepressant-like effects in mice.4 Behaves as an agonist at GPR55, EC50=39nM.5 Active in vivo.